Different receptor sites mediate opioid agonism and antagonism

J Med Chem. 1983 Oct;26(10):1341-3. doi: 10.1021/jm00364a001.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Binding Sites
  • Kinetics
  • Naltrexone / analogs & derivatives
  • Naltrexone / pharmacology
  • Narcotic Antagonists / pharmacology*
  • Narcotics / pharmacology*
  • Receptors, Opioid / drug effects
  • Receptors, Opioid / metabolism*
  • Structure-Activity Relationship

Substances

  • Narcotic Antagonists
  • Narcotics
  • Receptors, Opioid
  • Naltrexone
  • beta-funaltrexamine